[ 登录] [ 免费注册]
试剂仪器? title=
位置9a href="/">首页> 产品庒/a> > M-5011
立即咨询
咨询类型9/div>
*姓名9/div>
*电话9/div>
*单位9/div>
Email9/div>
*留言内容9/div>
请详细说明您的需求
*验证码:
M-5011
本产品不向个人销售,仅用作科学研究,不用于任何人体实验及非科研性质的动物实验、/div>
CAS NO: 76604-64-3
包装: 50mg, 100mg, 250mg
规格: ?8%

产品介绍

M-5011 is a non-steroidal anti-inflammatory drug and immunomodulator potentially for the treatment of inflammation and pain. M-5011 had an effective antinociceptive activity (ED50 value) of 0.63 mg/kg, being more potent than zaltoprofen (16.80 mg/kg) and tiaprofenic acid (4.78 mg/kg), equipotent to diclofenac sodium (0.68 mg/kg), and less potent than indomethacin (0.21 mg/kg) and ketoprofen (0.28 mg/kg). M-5011 partially inhibits the generalized bone loss accompanying the development of collagen-induced arthritis in rats. M-5011 is a useful NSAID that shows potent antinociceptive effects with low ulcerogenic activities. References: Horisawa E, Danjo K, Haruna M. Physical properties of solid dispersion of a nonsteroidal anti-inflammatory drug (M-5011) with Eudragit E. Drug Dev Ind Pharm. 2000 Dec;26(12):1271-8. PubMed PMID: 11147127.

纯度:≥98%

CAS?6604-64-3

Baidu
map