Binedaline, formerly known as Scha-1059, Ixprim, binodaline, is a drug that was being investigated as an antidepressant in the 1980s but never marketed. It acts as a selective norepinephrine reuptake inhibitor (Ki = 25 nM), with relatively insignificant influence on the serotonin (Ki = 847 nM) and dopamine (Ki >= 2 μM) transporters. It has negligible affinity for the α-adrenergic, mACh, H1, or 5-HT2 receptors. References: Saini T, Kumar S, Narasimhan B. Central Nervous System Activities of Indole Derivatives: An Overview. Cent Nerv Syst Agents Med Chem. 2015;16(1):19-28. Review. PubMed PMID: 26051466.

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CAS�?0662-16-0