Canniprene 是大麻独有的异戊二烯化联苄基,是 5-脂氧合酶 (
5-LO) 活 (
IC50=0.4 μM) 和环氧合?微粒体前列腺 E2 合酶 (
PGE2;
IC50=10 μM) 的有效抑制剂。Canniprene 抑制炎性类花生酸的产生并影响前列腺素的生成、/div>
| 生物活?/td> |
Canniprene, an isoprenylated bibenzyl unique toCannabis sativa, is a potent inhibitor of5-lipoxygenase(5-LO) activity (IC50=0.4 μM) and cyclooxygenase/microsomal prostaglandin E2 synthase (PGE2;IC50=10 μM). Canniprene inhibits the production of inflammatory eicosanoids and affects the generation of prostaglandins[1].
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| IC50& Target[1] |
5-LO 0.4 M (IC50) |
PGE2 10 M (IC50) |
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| 分子野/td> |
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| Formula |
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| CAS 叶/td> |
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| 中文名称 |
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| 结构分类 |
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| 来源 |
- Plants
- Moraceae
- Cannabis sativaL
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| 运输条件 |
Room temperature in continental US; may vary elsewhere.
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| 储存方式 |
Please store the product under the recommended conditions in the Certificate of Analysis.
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