| CAS: | 67469-81-2 | |
| 分子式: | C28H34N2O.2HCl | |
| 分子量: | 487.51 | |
| 英文名称: |
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| 用途: | GBR 12935双盐酸盐是多巴胺再吸收抑制剂。 |
| 货号 | 品牌 | 产品名称 | 规格 | 包装、参考价格 | |||||||||||||||||||||||||||||||||||||||
| G860914 | MACKLIN | GBR 12935双盐酸盐 | >98% | 384元/10mg; 720元/25mg; 1536元/100mg; 3520元/250mg; 6400元/500mg; | 咨询 | ||||||||||||||||||||||||||||||||||||||
储存:-20℃ 状态:灰白色到米黄色粉末 折射率:white solid | |||||||||||||||||||||||||||||||||||||||||||
| G9659 | Sigma-Aldrich | GBR 12935 dihydrochloride | ≥98% (TLC), powder | 2370.81元/25 MG; 8421.19元/100 MG; | 咨询 | ||||||||||||||||||||||||||||||||||||||
产品说明 应用 GBR 12935 dihydrochloride has been used as a dopamine reuptake inhibitor to study its effects on noradrenergic stimulation in the medial prefrontal cortex of rats (mPFC). It has also been used as a selective dopamine transporter (DAT) inhibitor to study its effects on behavior and neurochemical response in enriched condition (EC) and impoverished condition (IC) rats. 包装 25, 100 mg in poly bottle 生化/生理作用 GBR 12935 inhibits the dopamine and norepinephrine transporters with Kis of 21.5 nM and 225 nM, respectively. It does not inhibit the serotonin transporter (Ki = 6.5 mM). GBR 12935 binds to a nondopaminergic piperazine site in blood platelets and brain that has been identified as cytochrome P450. 特点和优势 This compound is featured on the Biogenic Amine Transporters page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here. 基本信息
产品性质
安全信息
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