CAS 56974-61-9; 甲磺酸加贝酯; 4-[[6-[(Aminoiminomethyl)amino]-1-oxohexyl]oxyl]benzoic acid ethyl ester mesylate salt

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货号

品牌

产品名称

规格

包装、参考价格

G864564

MACKLIN

Gabexate Mesylate

99%

29元/5mg; 30元/25mg; 49元/100mg; 198元/1g; 553元/5g;

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储存：-20°C
状态：白色固体

G798250

MACKLIN

Gabexate Mesylate

10mM in DMSO

907元/1ml;

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储存：-20°C

G0464

TCI

Gabexate Mesylate

>97.0%(N)

625元/1G;

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基本信息

纯度/分析方法	>97.0%(N)
分子式/分子量	C₁₆H₂₃N₃O₄・CH₄O₃S = 417.48
外观与形状(20℃)	固体
相关CAS RN	39492-01-8
Reaxys-RN	5702026
PubChem物质ID	253660880
Merck Index (14)	4320
MDL编号	MFCD00210299

技术规格

Appearance	White to Almost white powder to crystal
Purity(HPLC)	min. 94.0 area%
Purity(with Total Nitrogen)	min. 97.0 %
Melting point	89.0 to 93.0 ℃

物性(参考值)

熔点	91 ℃
水溶性	完全溶解
溶解性(易溶于)	氯仿,乙醇
溶解性(可溶于)	甲醇
溶解性(微溶于)	丙酮
溶解性(不溶于)	乙醚

相关法规

RTECS#

DG2800800

305432

J&K

Gabexate Mesylate

97%, 丝氨酸蛋白酶抑制剂

149元/1MG; 441元/5MG;

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基本信息

分子式	C₁₇H₂₇N₃O₇S
分子量	417.48
熔点	91
MDL编码	MFCD00210299
Beilstein	5702026
Merck	14,4320
存储条件	Freezer -20℃

安全信息

图形或危害标志
提示语	Warning
危险说明	H302 H410
防范说明	P264 P270 P273 P301+P312 P330 P391 P501
UN号码	3077
危险分类	9
包装等级	III
WGK	2
RTECS	DG2800800

SML2964

Sigma-Aldrich

Gabexate Mesylate

≥97% (HPLC)

841.96元/5 MG; 3400.25元/25 MG;

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产品说明

生化/生理作用

Gabexate mesylate is a competitive inhibitor of serine proteases that displays high selectivity for TMPRSS2 (Transmembrane protease serine 2) (IC50 = 130 nM) with little or no activity towards several MMPs, caspases and USPs (>> 10 μM). Gabexate mesylate was reported to decrease inflammatory cytokines production and be useful as an anticoagulant.

基本信息

经验(实验)分子式	C₁₆H₂₃N₃O₄ · CH₄O₃S
分子量	417.48
MDL编号	MFCD00210299

产品性质

质量水平	100
测定	≥97% (HPLC)
形式	powder
颜色	white to beige
溶解性	H₂O: 2 mg/mL, clear
储存温度	2-8℃
SMILES string	CS(O)(=O)=O.CCOC(=O)c1ccc(OC(=O)CCCCCNC(N)=N)cc1
InChI	1S/C16H23N3O4.CH4O3S/c1-2-22-15(21)12-7-9-13(10-8-12)23-14(20)6-4-3-5-11-19-16(17)18;1-5(2,3)4/h7-10H,2-6,11H2,1H3,(H4,17,18,19);1H3,(H,2,3,4)
InChI key	DNTNDFLIKUKKOC-UHFFFAOYSA-N

安全信息

储存分类代码	11 - Combustible Solids
WGK	WGK 2
闪点(F)	Not applicable
闪点(C)	Not applicable

G2417

Supelco

Gabexate Mesylate

analytical standard, for drug analysis

2946.73元/5 MG;

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产品说明

一般描述

Gabexate mesylate is a non-antigenic synthetic inhibitor of trypsin-like serine proteinases, which finds therapeutic applications in the treatment of disseminated intravascular coagulation and pancreatitis. It also plays the role of an anticoagulant in hemodialysis therapy.

应用

Refer to the product′s Certificate of Analysis for more information on a suitable instrument technique. Contact Technical Service for further support.

包装

5 mg in glass bottle

基本信息

经验(实验)分子式	C₁₆H₂₃N₃O₄ · CH₄O₃S
分子量	417.48
MDL编号	MFCD00210299
PubChem化学物质编号	329799903
NACRES	NA.24

产品性质

质量水平	200
等级	analytical standard, for drug analysis
形式	solid
technique(s)	HPLC: suitable gas chromatography (GC): suitable
application(s)	forensics and toxicology pharmaceutical (small molecule) veterinary
格式	neat
SMILES string	CS(O)(=O)=O.CCOC(=O)c1ccc(OC(=O)CCCCCNC(N)=N)cc1
InChI	1S/C16H23N3O4.CH4O3S/c1-2-22-15(21)12-7-9-13(10-8-12)23-14(20)6-4-3-5-11-19-16(17)18;1-5(2,3)4/h7-10H,2-6,11H2,1H3,(H4,17,18,19);1H3,(H,2,3,4)
InChI key	DNTNDFLIKUKKOC-UHFFFAOYSA-N

安全信息

储存分类代码	11 - Combustible Solids
WGK	WGK 2
闪点(F)	Not applicable
闪点(C)	Not applicable
个人防护装备	Eyeshields, Gloves, type N95 (US)