| CAS: | 371980-98-2 | ||
| 分子式: | C24H29Cl2NO · HCl | ||
| 分子量: | 454.86 | ||
| 英文名称: |
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| 用途: | SB-612111 is a potent antagonist of the nociceptin receptor ORL-1. SB-612111 binds to ORL-1 with high affinity (Ki = 0.33 nM) but has very low affinity for classic opioid receptors. The compound SB-612111 antagonizes the anti-morphine effects of nociceptin and blocks nociceptin-induced thermal hyperalgesia. |
| 货号 | 品牌 | 产品名称 | 规格 | 包装、参考价格 | |||||||||||||||||||||||||||||
| S921012 | MACKLIN | SB-612111 hydrochloride | ≥98% (HPLC) | 1048元/5mg; | 咨询 | ||||||||||||||||||||||||||||
储存:−20°C 状态:固体 | |||||||||||||||||||||||||||||||||
| SML0571 | Sigma-Aldrich | SB-612111 hydrochloride | ≥98% (HPLC) | 1549.77元/5 MG; 6268.49元/25 MG; | 咨询 | ||||||||||||||||||||||||||||
产品说明 包装 5, 25 mg in glass bottle 生化/生理作用 SB-612111 is a potent antagonist of the nociceptin receptor ORL-1. SB-612111 binds to ORL-1 with high affinity (Ki = 0.33 nM) but has very low affinity for classic opioid receptors. The compound SB-612111 antagonizes the anti-morphine effects of nociceptin and blocks nociceptin-induced thermal hyperalgesia. 特点和优势 This compound is featured on the Opioid Receptors page of the Handbook of Receptor Classification and Signal Transduction. To browse other handbook pages, click here. 基本信息
产品性质
安全信息
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